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Efficient One-Pot Synthesis (efficient + one-pot_synthesis)
Selected AbstractsA Facile and Efficient One-Pot Synthesis of Substituted Quinolines from ,-Arylamino Ketones Under Vilsmeier ConditionsEUROPEAN JOURNAL OF ORGANIC CHEMISTRY, Issue 24 2009Yan Wang Abstract An efficient one-pot synthesis of substituted quinolines from ,-arylamino ketones in the presence of PBr3 in DMF has been developed. This general protocol provides a novel and facile access to substituted quinolines by sequential Vilsmeier,Haack reaction, intramolecular cyclization and aromatization reactions of ,-arylamino ketones. PBr3 plays a dual role in the quinoline synthesis: as a key component of the Vilsmeier reagent (PBr3/DMF) and as a reducing reagent. (© Wiley-VCH Verlag GmbH & Co. KGaA, 69451 Weinheim, Germany, 2009) [source] Highly Efficient One-Pot Synthesis of 2-Substituted Quinazolines and 4H -Benzo[d][1,3]oxazines via Cross Dehydrogenative Coupling using Sodium HypochloriteADVANCED SYNTHESIS & CATALYSIS (PREVIOUSLY: JOURNAL FUER PRAKTISCHE CHEMIE), Issue 2-3 2010C. Uma Maheswari Abstract This communication describes a catalyst-free synthesis of 2-substituted quinazolines and 4H -benzo[d][1,3]oxazines using commericially available sodium hypochlorite as oxidant. Operational simplicity, mild reaction conditions and the ability to construct structurally diverse 2-quinazolines and 2-substituted 4H -benzo[d][1,3]oxazines by this method render it to be a practical alternative for the synthesis of these heterocycles. [source] ChemInform Abstract: An Efficient One-Pot Synthesis of Trifluoromethyl-Substituted Cyclobutene Derivatives.CHEMINFORM, Issue 38 2010Mohmmad Hossein Mosslemin Abstract Cyclobutene derivatives (III) are obtained via intramolecular Wittig reaction between 1,1,1-trifluorobutane-2,4-diones and ethyl phenylpropiolate. [source] ChemInform Abstract: Efficient One-Pot Synthesis of 6-Arylpyrrolo[3,2-d]pyrimidines from 6-Arylethynyl-5-nitropyrimidines.CHEMINFORM, Issue 36 2010Inga Cikotiene Abstract The synthesis of the biologically important heterocyclic system involves conjugative addition of diethylamine to ethynylpyrimidines (I) and subsequent reductive cyclization. [source] ChemInform Abstract: An Efficient One-Pot Synthesis of 3-Aryl-1,2,4-oxadiazol-5-amines under Solvent-Free Conditions.CHEMINFORM, Issue 25 2010Mehdi Adib Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: Efficient One-Pot Synthesis of Spirooxindole Derivatives by Ethylenediamine Diacetate Catalyzed Reactions in Water.CHEMINFORM, Issue 23 2010Galla Sri Hari Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: Efficient One-Pot Synthesis of 2,4-Di(het)aryl and 2,4-Diamino Pyrido[3,2-d]pyrimidines Involving Regioselective SNAr and Palladium-Catalyzed Reactions.CHEMINFORM, Issue 18 2010Abdellatif Tikad Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: An Efficient One-Pot Synthesis of Naphthoxazinones by a Three-Component Coupling of Naphthol, Aldehydes, and Urea Catalyzed by Zinc Triflate.CHEMINFORM, Issue 6 2010Alakananda Hajra Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: A Novel Three-Component Reaction of a Secondary Amine and a 2-Hydroxybenzaldehyde Derivative with an Isocyanide in the Presence of Silica Gel: An Efficient One-Pot Synthesis of Benzo[b]furan Derivatives.CHEMINFORM, Issue 2 2010Ali Ramazani Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: A Safe, Convenient and Efficient One-Pot Synthesis of ,-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride.CHEMINFORM, Issue 49 2009Jun Yu Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: Efficient One-Pot Synthesis of 4-EthynylbenzenesulfonamidesCHEMINFORM, Issue 30 2009Wensheng Zhang Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: ZrCl4 Promoted Efficient One-Pot Synthesis of ,-Amino Nitriles.CHEMINFORM, Issue 24 2009M. Raghu Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: Efficient One-Pot Synthesis of Hydroxyflavanones by Cyclization and O-Demethylation of Methoxychalcones.CHEMINFORM, Issue 45 2008Tao Liu Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: An Efficient One-Pot Synthesis of Tethered Cyclohexadiene Enaminonitriles from Methyl-Ketones: An Effective Route to Quinazolines.CHEMINFORM, Issue 42 2008Bennie J. Bench Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: An Efficient One-Pot Synthesis of 3-Substituted-5-amino-1,2,4-thiadiazoles from Isothiocyanates and Amidines.CHEMINFORM, Issue 33 2008Yong-Jin Wu Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: Efficient One-Pot Synthesis of Polyfunctionalized Thiophenes via an Amine-Mediated Ring Opening of EWG-Activated 2-Methylene-1,3-dithioles.CHEMINFORM, Issue 14 2008Fushun Liang Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] Indium Trichloride Catalyzed Efficient One-Pot Synthesis of Highly Substituted Furans.CHEMINFORM, Issue 29 2007Sumit Dey Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF. [source] An Efficient One-Pot Synthesis of Polyhydrobenzoacridine-1-one Derivatives under Microwave Irradiation Without Catalyst.CHEMINFORM, Issue 13 2007Shujiang Tu Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF. [source] Confirmation and Prevention of Halogen Exchange: Practical and Highly Efficient One-Pot Synthesis of Dibromo- and Dichloropyridazinones.CHEMINFORM, Issue 13 2007Ji Zhang Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF. [source] Reaction Between Phosphines and Itaconic Anhydride in the Presence of Water: An Efficient One-Pot Synthesis of 5-Oxo-1,2,5 -oxaphospholanes.CHEMINFORM, Issue 29 2006Mohammad Bagher Teimouri Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF. [source] An Efficient One-Pot Synthesis of 3-(2-Oxo-2H-chromen-3-yl)-6H,8H-pyrimido[4,5-c]pyridazine-5,7-diones.CHEMINFORM, Issue 4 2006V. Rajeswar Rao No abstract is available for this article. [source] An Efficient One-Pot Synthesis of Aminobenzimidazoles.CHEMINFORM, Issue 20 2005David M. D. Fouchard Abstract For Abstract see ChemInform Abstract in Full Text. [source] An Efficient One-Pot Synthesis of Annulated Pyridines Utilizing a Directed ortho-Metalation/Transmetalation Approach.CHEMINFORM, Issue 23 2004Antony J. Davies Abstract For Abstract see ChemInform Abstract in Full Text. [source] An Efficient One-Pot Synthesis of 2-Hydroxyalkyl Dithiocarbamates.CHEMINFORM, Issue 42 2003Jia-ling Cui Abstract For Abstract see ChemInform Abstract in Full Text. [source] An Efficient One-Pot Synthesis of 6-Alkoxy-8,9-dialkylpurines via Reaction of 5-Amino-4-chloro-6-alkylaminopyrimidines with N,N-Dimethylalkaneamides and Alkoxide Ions.CHEMINFORM, Issue 1 2003Pier Giovanni Baraldi Abstract For Abstract see ChemInform Abstract in Full Text. [source] An Efficient One-Pot Synthesis of Carbamate Esters Through Alcoholic Tosylates.CHEMINFORM, Issue 50 2002Devdutt Chaturvedi No abstract is available for this article. [source] ChemInform Abstract: Microwave-Assisted Efficient One-Pot Synthesis of Nitriles in Dry Media.CHEMINFORM, Issue 45 2001J. S. Yadav Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] ChemInform Abstract: An Efficient One-Pot Synthesis of Functionalized Azamacrocycles from Methyl 2-Siloxy-2-vinylcyclopropanecarboxylates.CHEMINFORM, Issue 17 2001Pranab K. Patra Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a "Full Text" option. The original article is trackable via the "References" option. [source] A Facile and Efficient One-Pot Synthesis of Substituted Quinolines from ,-Arylamino Ketones Under Vilsmeier ConditionsEUROPEAN JOURNAL OF ORGANIC CHEMISTRY, Issue 24 2009Yan Wang Abstract An efficient one-pot synthesis of substituted quinolines from ,-arylamino ketones in the presence of PBr3 in DMF has been developed. This general protocol provides a novel and facile access to substituted quinolines by sequential Vilsmeier,Haack reaction, intramolecular cyclization and aromatization reactions of ,-arylamino ketones. PBr3 plays a dual role in the quinoline synthesis: as a key component of the Vilsmeier reagent (PBr3/DMF) and as a reducing reagent. (© Wiley-VCH Verlag GmbH & Co. KGaA, 69451 Weinheim, Germany, 2009) [source] Highly Efficient Ligands for the Palladium-Assisted Double N -Arylation of Primary Amines for One-Sep Construction of CarbazolesADVANCED SYNTHESIS & CATALYSIS (PREVIOUSLY: JOURNAL FUER PRAKTISCHE CHEMIE), Issue 4 2010Yibo Zhou Abstract A highly efficient one-pot synthesis of carbazoles via palladium-catalyzed double N -arylation of primary amines with 2,2,-dihalobiphenyls is described using a catalyst system comprised of tris(dibenzylideneacetone)dipalladium(0) (Pd2dba3) and the proazaphosphatrane P(i -BuNCH2CH2)3N (8) or its derivative (t- Bu)2PNP(i- BuNCH2CH2)3N (9a) as the ligand. The process is effective for double N -arylation of 2,2,-biphenyl dibromide, diiodide, and even dichloride with a variety of primary amines including neutral, electron-rich, electron-deficient, and sterically hindered anilines as well as aliphatic amines. [source] |